Velagliflozin |
Last updated: 18/10/2024 |
(Not known by any other names) |
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An antidiabetic veterinary medication | |
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Current | |
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Used to manage Diabetes mellitus helping to reduce hyperinsulinemia and insulin resistance | |
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Cats; Horses; Ponies |
Approval status |
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Approved | |
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Approved |
Chemical structure |
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Isomeric | |
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C₂₃H₂₅NO₅ | |
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C1CC1C2=CC=C(C=C2)CC3=C(C=CC(=C3)C4C(C(C(C(O4)CO)O)O)O)C#N | |
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C1CC1C2=CC=C(C=C2)CC3=C(C=CC(=C3)[C@H]4[C@@H]([C@H]([C@@H]([C@H](O4)CO)O)O)O)C#N | |
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SENUNDCNOYAWGN-ZQGJOIPISA-N | |
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InChI=1S/C23H25NO5/c24-11-17-8-7-16(23-22(28)21(27)20(26)19(12-25)29-23)10-18(17)9-13-1-3-14(4-2-13)15-5-6-15/h1-4,7-8,10,15,19-23,25-28H,5-6,9,12H2/t19-,20-,21+,22-,23+/m1/s1 | |
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Yes |
General status |
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Medicinal drug; Antidiabetic medication | |
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Unclassified veterinary drug | |
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95% | |
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Synthetic | |
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Sodium-glucose co-transporter2 inhibior | |
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[Sodium-glucose cotransporter 2, Inhibitor] | |
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946525-65-1 | |
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24862817 | |
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Alimentary tract and metabolism: Sodium-glucose co-transporter 2 inhibitors | |
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QA10BK90 | |
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No | |
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395.4 | |
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2-[(4-cyclopropylphenyl)methyl]-4-[(2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]benzonitrile | |
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2-[(4-cyclopropylphenyl)methyl]-4-[(2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]benzonitrile | |
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Off-white coloured solid |
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Senvelgo oral solution | Boehringer Ingelheim Animal Health UK | GB National authorisation | Prescription only medicine to be authorised by a veterinarian (POM-V) | ||||||
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Usually supplied as an oral solution |
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648.6 | Q3 Q = Miscellaneous data from online sources 3 = Unverified data of known source |
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346.1 | Q3 Q = Miscellaneous data from online sources 3 = Unverified data of known source |
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6.61 X 1003 | Calculated | - | |||||||
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3.82 | Q3 Q = Miscellaneous data from online sources 3 = Unverified data of known source |
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1.39 | Q3 Q = Miscellaneous data from online sources 3 = Unverified data of known source |
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1.67 | Q3 Q = Miscellaneous data from online sources 3 = Unverified data of known source |
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Degradation |
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As this parameter is not normally measured directly, a surrogate measure is used: ‘Photochemical oxidative DT₅₀’. Where data is available, this can be found in the Fate Indices section below. | ||||||||||
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Soil adsorption and mobility |
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Fate indices |
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Known metabolites |
None
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Terrestrial ecotoxicology |
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Aquatic ecotoxicology |
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General |
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Eliminated unchanged in faeces in around 7 hrs | Q3 Q = Miscellaneous data from online sources 3 = Unverified data of known source |
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Health issues |
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No information available |
Handling issues |
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Avoid dust generation | |||
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Health: H335, H319, H315 | |||
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Not listed (Not listed) | |||
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Not regulated | |||
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Shelf-life as packaged is 3 yrs. 6 months once opened. Generally stable. |
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velagliflozin | ||
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Record last updated: | 18/10/2024 |
Contact: | aeru@herts.ac.uk |
Please cite as: | Lewis, K.A., Tzilivakis, J., Warner, D. and Green, A. (2016) An international database for pesticide risk assessments and management. Human and Ecological Risk Assessment: An International Journal, 22(4), 1050-1064. DOI: 10.1080/10807039.2015.1133242 |