Epinephrine acid tartrate |
Last updated: 23/05/2024 |
(Also known as: (-)-epinephrine bitartrate; adrenaline bitartrate) |
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Epinephrine is widely used drug for anaphylactoid shock | |
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Current | |
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Primarily used to treat anaphylaxis and for cardiac resuscitation | |
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Dogs; Cats; Other domesticated animals; Cattle; Horses; Pigs; Sheep |
Approval status |
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Approved | |
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Approved |
Chemical structure |
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Isomeric. The R-enantiomer of epinephrine is the hormone secreted by the adrenal glands. | |
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C₁₃H₁₉NO₉ | |
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CNCC(C1=CC(=C(C=C1)O)O)O.C(C(C(=O)O)O)(C(=O)O)O | |
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CNC[C@@H](C1=CC(=C(C=C1)O)O)O.C(C(C(=O)O)O)(C(=O)O)O | |
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YLXIPWWIOISBDD-FVGYRXGTSA-N | |
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InChI=1S/C9H13NO3.C4H6O6/c1-10-5-9(13)6-2-3-7(11)8(12)4-6;5-1(3(7)8)2(6)4(9)10/h2-4,9-13H,5H2,1H3;1-2,5-6H,(H,7,8)(H,9,10)/t9-;/m0./s1 | |
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Yes |
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Common Name | Relationship | Link |
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epinephrine | Parent |
General status |
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Medicinal drug | |
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Hormone | |
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Unclassified medicinal drug; Hornone | |
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Synthetic | |
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Antagonizes the effects of histamine, raises blood sugar, increases heart rate and contractility, and increases systolic blood pressure. | |
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[Adrenergic receptors] | |
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51-42-3 | |
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200-097-1 | |
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6852374 | |
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Multiple therapeutic classes | |
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QA01AD01; QB02BC09; QC01CA03; QC01CA24; QR01AA14; QR03AA01; QR03AK01; QS01EA01; QS01EA51 | |
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No | |
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333.29 | |
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2,3-dihydroxybutanedioic acid;4-[(1R)-1-hydroxy-2-(methylamino)ethyl]benzene-1,2-diol | |
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Formulations |
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Lignol Solution for Injection | Dechra Limited | UK National authorisation | Prescription only medicine to be authorised by suitably qualified person (POM-VPS) | ||||||
Procamidor Duo 40 mg/ml + 0.036 mg/ml Solution for Injection | VetViva Richter GmbH | GB National authorisation | Prescription only medicine to be authorised by suitably qualified person (POM-VPS) | |||||||
Pronestesic 40 mg/ml / 0.036 mg/ml Solution for Injection | Fatro S.p.A. | GB National authorisation | Prescription only medicine to be authorised by a veterinarian (POM-V) | |||||||
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Usually formulated as solutions for injection but also as cutaneous sprays for topical use |
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As this parameter is not normally measured directly, a surrogate measure is used: ‘Photochemical oxidative DT₅₀’. Where data is available, this can be found in the Fate Indices section below. | ||||||||||
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Soil adsorption and mobility |
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Fate indices |
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Known metabolites |
None
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Terrestrial ecotoxicology |
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90 | Q3 Q = Miscellaneous data from online sources Mouse3 = Unverified data of known source |
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General |
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90 | Q3 Q = Miscellaneous data from online sources Mouse3 = Unverified data of known source |
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Excreted rapidly in urine | Q3 Q = Miscellaneous data from online sources 3 = Unverified data of known source |
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Health issues |
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No information available |
Handling issues |
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When heated to decomposition it will emit toxic fumes Combustible IMDG Transport Hazard Class 6.1 |
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Health: H301, H311, H315, H319, H335 | |||
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Not listed (Not listed) | |||
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UN2811 | |||
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Packaging Group II (moderate danger) | |||
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Chemically stable under standard ambient conditions |
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epinephrine acid tartrate | ||
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Record last updated: | 23/05/2024 |
Contact: | aeru@herts.ac.uk |
Please cite as: | Lewis, K.A., Tzilivakis, J., Warner, D. and Green, A. (2016) An international database for pesticide risk assessments and management. Human and Ecological Risk Assessment: An International Journal, 22(4), 1050-1064. DOI: 10.1080/10807039.2015.1133242 |