Fentanyl citrate |
Last updated: 22/05/2024 |
(Not known by any other names) |
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A potent class-II opiate narcotic veterinary medication | |
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Current | |
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1960, first synthesised | |
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Mainly used as a sedative or tranquilizer for various veterinary surgical procedures and for severe pain management | |
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Sheep; Goats; Dogs; Cats; Bears; Pigs; Rats; Mice; Rabbits |
Approval status |
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Approved | |
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Approved |
Chemical structure |
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- | |
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C₂₈H₃₆N₂O₈ | |
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CCC(=O)N(C1CCN(CC1)CCC2=CC=CC=C2)C3=CC=CC=C3.C(C(=O)O)C(CC(=O)O)(C(=O)O)O | |
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IVLVTNPOHDFFCJ-UHFFFAOYSA-N | |
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InChI=1S/C22H28N2O.C6H8O7/c1-2-22(25)24(20-11-7-4-8-12-20)21-14-17-23(18-15-21)16-13-19-9-5-3-6-10-19;7-3(8)1-6(13,5(11)12)2-4(9)10/h3-12,21H,2,13-18H2,1H3;13H,1-2H2,(H,7,8)(H,9,10)(H,11,12) | |
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Yes |
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Common Name | Relationship | Link |
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fentanyl citrate | - | |
fentanyl citrate hydrate | Hydrate | |
fentanyl | Parent |
General status |
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Analgesic, Anesthetic, Medicinal drug | |
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Synthetic opioid | |
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Synthetic | |
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A mu-opioid agonist | |
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[Mu-type opioid receptor, Agonist], [Delta-type opioid receptor, agonist], [Kappa-type opioid receptor, Agonist] | |
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990-73-8 | |
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213-588-0 | |
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13810 | |
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Nervous system: Anesthetics | |
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QN01AH51 | |
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UK: Class A, Schedule 2; EU: UN61/72, Class I | |
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528.6 | |
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2-hydroxypropane-1,2,3-tricarboxylic acid;N-phenyl-N-[1-(2-phenylethyl)piperidin-4-yl]propanamide | |
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- | |
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USA Superlist DEA Schedule II | |
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Formulations |
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Hypnorm Solution for Injection | Animal Medics UK Ltd | UK National authorisation | Prescription only medicine to be authorised by a veterinarian (POM-V) | ||||||
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Usually formulated as solutions for injection |
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As this parameter is not normally measured directly, a surrogate measure is used: ‘Photochemical oxidative DT₅₀’. Where data is available, this can be found in the Fate Indices section below. | ||||||||||
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Fate indices |
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Known metabolites |
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Terrestrial ecotoxicology |
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3.1 | F4 F = U.S. EPA ECOTOX database / U.S. EPA pesticide fate database / Miscellaneous WHO documents / FAO data, IPCS INCHEM data (US EPA Databases Related to Pesticide Risk Assessment ) Rat4 = Verified data |
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Aquatic ecotoxicology |
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General |
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High (class III) | - | - | ||||||||
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3.1 | F4 F = U.S. EPA ECOTOX database / U.S. EPA pesticide fate database / Miscellaneous WHO documents / FAO data, IPCS INCHEM data (US EPA Databases Related to Pesticide Risk Assessment ) Rat4 = Verified data |
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May be absorbed through dermal contact | ||||||||||
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Considerable metabolism, up to 75% excreted as metabolites in the urine, less lost via the faeces, <10% unchanged | F4 F = U.S. EPA ECOTOX database / U.S. EPA pesticide fate database / Miscellaneous WHO documents / FAO data, IPCS INCHEM data (US EPA Databases Related to Pesticide Risk Assessment ) 4 = Verified data |
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Health issues |
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May cause diarrhoea, nausea, constipation, dry mouth, somnolence and confusion May cause respiratory depression |
Handling issues |
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No information available | |||
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Not listed (Not listed) | |||
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fentanyl citrate | ||
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fentanila | ||
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Record last updated: | 22/05/2024 |
Contact: | aeru@herts.ac.uk |
Please cite as: | Lewis, K.A., Tzilivakis, J., Warner, D. and Green, A. (2016) An international database for pesticide risk assessments and management. Human and Ecological Risk Assessment: An International Journal, 22(4), 1050-1064. DOI: 10.1080/10807039.2015.1133242 |